
ọja Apejuwe
Peony glycosides funfun jẹ monoterpene glycoside ti a fa jade lati awọn gbongbo Paeonia lactiflora, ti a mọ gẹgẹ bi eroja pataki ti oogun Kannada ibile "White Peony Root" pẹlu ifihan atako - iredodo, analgesic, ati awọn ipa aiṣedeede neuroprotective. Lilo imọ-ẹrọ isọdọmọ giga{2}}iyara - lọwọlọwọ chromatography (HSCCC), ọja wa ṣaṣeyọri aṣeyọri kan 99.5% ultra{5}mimọ giga pẹlu 5× imudara bioavailability ni akawe si awọn iyọkuro ti aṣa. Akojọ si bi boṣewa itọkasi ni Kannada Pharmacopoeia 2020.
Ọja eroja
|
Paramita |
Awọn pato |
|
Orisun |
Si dahùn o wá tiPaeonia lactifloraPall. (Ranunculaceae) |
|
Ifarahan |
Funfun lati pa- lulú kristali funfun |
|
Mimo |
Ti o tobi ju tabi dọgba si 98% (HPLC) |
|
Fọọmu Molecular |
C₂₃H₂₈O₁₁ |
|
Òṣuwọn Molikula |
480.47 |
|
Solubility |
Tiotuka larọwọto ni methanol/ethanol, tiotuka die ninu omi (1g/100mL, iwọn 25) |
|
Awọn iwe-ẹri |
ISO22000, HACCP, USDA Organic, Halal |
Imọ Tiwqn Analysis
|
Ẹya ara ẹrọ |
Akoonu/Properties |
Awọn anfani |
|
Paeoniflorin |
Ti o tobi ju tabi dọgba si 98% (HPLC-ELSD) |
NF{{0}κB idinamọ ipa ọna (30% munadoko diẹ sii ju dexamethasone) |
|
Albiflorin |
Kere ju tabi dọgba si 1.0% |
Iṣiṣẹpọ ni imudara iṣẹ ṣiṣe olugba GABA (anxiolytic) |
|
Awọn Irin Eru |
Pb Kere ju tabi dogba si 0.5ppm |
Ni ibamu pẹlu ICH Q3D awọn itọsona aimọ alaimọ |
|
Awọn iṣẹku ti o yanju |
Methanol Kere ju tabi dogba si 200ppm |
Pade awọn ibeere EP pharmacopeia |
Awọn paramita bọtini:
Ojuami Iyo: 196-198 ìyí (ibajẹ)
Yiyi pato: [ ]D²⁰=-12.5 ìyí (c=1, ninu methanol)
Isonu lori GbigbeKere ju tabi dogba si 1.0%
Awọn ohun elo
▍ Awọn oogun oogun
Anti-Abẹrẹ inu Arthritis: Ni idapọ pẹlu methotrexate (majele ti dinku)
NeuroprotectantsAwọn agbekalẹ Ischemic stroke IV (Awọn idanwo Ipele III)
▍ Nutraceuticals
Idaabobo ẸdọDinku awọn ipele ALT/AST dinku (40% dinku ninu awọn idanwo ile-iwosan)
Atako -Abanuje Gummies: Iyara - itusilẹ (ibẹrẹ iṣẹju 15)
▍ Ohun ikunra
Titunṣe Awọ Awọ: Idinamọ olugba TRPV1 (72% ↓ sisun sisun)
Atako -Omi Irun Irun: Ṣe afikun ipele anagen (35% ↑ iwuwo irun ni vivo)
▍ Oogun Ogbo
Ijapa Alapapọ: Dinku iwọn lilo phenobarbital nipasẹ 30%
▍ Iwadi Reagents
TLR4 ipa ọna StudiesIwọn ayẹwo sẹẹli (CAS 23180-57-6)
Iṣakojọpọ & Ibi ipamọ
- Iṣakojọpọ: 1kg / apo bankanje, 25kg / ilu okun (afaraṣe)
- Ibi ipamọ: Itaja ni itura kan, ibi gbigbẹ, edidi ati aabo lati ina
- Igbesi aye selifu: Awọn oṣu 24 (labẹ awọn ipo ṣiṣi silẹ)

Ọkan Duro iṣẹ
Ohun elo Raw → Powder → Jade → Awọn ọja OEM ti pari
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